• Title/Summary/Keyword: R-maps

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Design of the New Insecticidal Active Molecule against Diamond-Back Moth (Plutella Xylostella Linnaeus) (배추좀나방(Plutella Xylostella Linnaeus)에 대한 새로운 살충활성 분자의 설계)

  • Cho, Yun-Gi;Choi, Woo-Young;Sung, Nack-Do
    • Korean Journal of Agricultural Science
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    • v.34 no.2
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    • pp.171-179
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    • 2007
  • The new insecticidal active molecules from the based on the holographic quantitative structure-activity relationships (HQSAR) between a series of $1-(R_1)-2-(n-octyl)-3-(R_2)$, $3-(R_3)-pseudothiourea$ derivatives and their insecticidal activities against Diamond-back moth (Plutella Xylostella Linnaeus) were designed and discussed quantitatively. The most active molecule from the based graphical analyses of atomic contribution maps with the optimized HQSAR C-1 model ($q^2=0.764$ & $r^2{ncv}=0.942$) was 1-(n-butyl)-2-(t-butyl)-3,3-diisopropylpseudothiourea (P1: $pI_{50}=5.30$, $IC_{50}=1.397ppm$). Therefore, it is suggested that the new designed molecule would increased the activity as much as 23.5 times as compared to X=n-octyl substituent 17($pI_{50}=4.00$, $IC_{50}=32.86ppm$) which was the highest active molecule in training set compounds.

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Molecular Holographic QSAR Model on the Herbicidal Activities of New Novel 2-(4-(6-chloro-2-benzoxazolyloxy)phenoxy)-N-phenylpropionamide Derivatives and Prediction of Higher Activity Compounds (새로운 2-(4-(6-chloro-2-benzoxazolyloxy)phenoxy)-N-phenyl-propionamide 유도체들의 제초활성에 관한 HQSAR 모델과 높은 활성 화합물의 예측)

  • Sung, Nack-Do;Kim, Dae-Whang;Jung, Hoon-Sung
    • The Korean Journal of Pesticide Science
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    • v.9 no.4
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    • pp.279-286
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    • 2005
  • The herbicidal activities against pre-emergence barnyard grass (Echinochloa crus-galli) by a series of new 2-(4-(6-chloro-2-benzoxazolyloxy)phenoxy)-N-phenylpopionamide derivatives as substrate molecule were studied using molecular holographic (H) quantitative structure activity relationships (HQSAR) methodology. From the based on the findings, the higher herbicidal active compounds are predicted by the derived HQSAR model. The best HQSAR model (VI-1) was derived from fragment distinction combination of atoms/bonds in fragment size, $7{\sim}10$bin. The herbicidal activities from atomic contribution maps showed that the activity will be able to increased according to the R-substituents variation of the N-phenyl ring and change of 6-chloro-2-benzoxazolyloxy group. Based on the results, the statistical results of the best HQSAR model (VI-1) exhibited the best pedictability and fitness for the herbicidal activities based on the cross-validated value ($q^2=0.646$) and non cross-validated value ($r^2_{ncv.}=0.917$), respectively. From the graphical analyses of atomic contribution maps, it was revealed that the lowest herbicidal activitics depends upon the 4-(6-chloro-2-benzoxazolyloxy)phenoxy group ($pred.pI_{50}=-3.20$). Particularly, the R=4-fluoro, X=isobutoxy substituent (P2) of (X)-phenoxy-N-(R)-phenylpropionamide derivative is predicted as the highest active compound ($pred.pI_{50}=9.12$).

SUBSTITUTION OPERATORS IN THE SPACES OF FUNCTIONS OF BOUNDED VARIATION BV2α(I)

  • Aziz, Wadie;Guerrero, Jose Atilio;Merentes, Nelson
    • Bulletin of the Korean Mathematical Society
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    • v.52 no.2
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    • pp.649-659
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    • 2015
  • The space $BV^2_{\alpha}(I)$ of all the real functions defined on interval $I=[a,b]{\subset}\mathbb{R}$, which are of bounded second ${\alpha}$-variation (in the sense De la Vall$\acute{e}$ Poussin) on I forms a Banach space. In this space we define an operator of substitution H generated by a function $h:I{\times}\mathbb{R}{\rightarrow}\mathbb{R}$, and prove, in particular, that if H maps $BV^2_{\alpha}(I)$ into itself and is globally Lipschitz or uniformly continuous, then h is an affine function with respect to the second variable.

Optimal Depth Calibration for KinectTM Sensors via an Experimental Design Method (실험 계획법에 기반한 키넥트 센서의 최적 깊이 캘리브레이션 방법)

  • Park, Jae-Han;Bae, Ji-Hum;Baeg, Moon-Hong
    • Journal of Institute of Control, Robotics and Systems
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    • v.21 no.11
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    • pp.1003-1007
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    • 2015
  • Depth calibration is a procedure for finding the conversion function that maps disparity data from a depth-sensing camera to actual distance information. In this paper, we present an optimal depth calibration method for Kinect$^{TM}$ sensors based on an experimental design and convex optimization. The proposed method, which utilizes multiple measurements from only two points, suggests a simplified calibration procedure. The confidence ellipsoids obtained from a series of simulations confirm that a simpler procedure produces a more reliable calibration function.

Isolation and characterization of corynebacteria-E. coli shuttle vector pKU6 from coryneform bacteria (Corynebacteria-E. coli shuttle vector pKU6의 분리 및 확인)

  • 허태린;이진우;이세영
    • Korean Journal of Microbiology
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    • v.22 no.4
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    • pp.249-255
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    • 1984
  • To develop the host-vector system for industrial Coryneform bacteria that seemed to be the most suitable microorganisms for molecular breeding of genes involved in the production of amion acids, nucleotides, and other products of industrial interest, broad host range E. coli plasmid R 1162 DNA was transformed into Brevibacterium ammoniagenes and the plasmids pKU6 isolated from a transformant was physically characterized. All other plasmids from the transformed cells except pKU6 exsisted as multimeric forms in Brevibacterium ammoniagenes. The plasmid DNA was retransformed into Corynebacterium glutamicum with a high frequency ($1.32{\times}10^{-1}$ per cell) and maintained stably both in Brevibacterium ammoniagenes and Corynebacterium glutamicum after 100 generations of cultures with 25-30 copy number per cell. The size of both plasmid pKU6 and plasmid R1162 were the same and restriction maps by EcoR I, Ava I, Pst I, Pvu II and Hinc II were also similar.

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Metadata Design Based on Vector Type Geospatial Information Standard for the Collection and Management of Inundation Map (침수지도 수집 및 관리를 위한 벡터형 공간정보 표준 기반의 메타데이터 설계)

  • Sim, Gyu-Seong
    • Journal of the Korea Academia-Industrial cooperation Society
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    • v.17 no.5
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    • pp.42-48
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    • 2016
  • Inundation Maps are used to predict potential areas of flooding through the signs of past flooding and flood inundation analysis for flooding expected in the future, and this has led to the development of various forms of disaster-related services by governments. However, each institution has its own individual scenarios for making maps for spatial expression. Therefore, the type of spatial information is not standardized and has many forms and structures. In this study, we attempted to design the metadata that would allow Inundation Map information to be shared and used in various fields. The international standard, ISO 19115, and the domestic standards, KS X ISO 19115, TTAS.IS - 19115 and TTAS.KO - 10.0139/R1 of TTA, were used in the design to derive an appropriate standard for comparative analysis by dividing into maintenance, constraints, metadata, spatial reference system, identification, and distribution. It is expected that inundation maps will be easier to utilize and distribute among institutions and private companies by systematically collecting and managing them through the metadata design based vector space information standard developed in this study.

Analysis of Current Situation and Relationship among National R&D Projects for Technology Convergence (국가 융합연구사업의 현황 및 연계성 분석)

  • Cho, Yangrae;Yang, Iesuk;Suh, Yongyoon;Jeon, Jeonghwan
    • Journal of Korean Institute of Industrial Engineers
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    • v.41 no.3
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    • pp.305-323
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    • 2015
  • Since various R&D projects about technology convergence was conducted by the government of Korea, the lack of liaisons among the projects has been accepted as serious issues related on the duplicated funding. In this article, we propose a research framework to analyze the relationship among national R&D projects about technology convergence. In detail, the projects have been sorted and categorized with the data collected from National Science and Technology Information Service (NTIS) in order to analyze the current state of national R&D projects. The linkages among projects are then established using the results of analysis on national R&D projects. Finally, the relationship maps have been developed. It is expected that the result could be applied to identify the relations among projects and handle problems on the duplicated funding.

TOPOLOGIES AND INCIDENCE STRUCTURE ON Rn-GEOMETRIES

  • Im, Jang-Hwan
    • Journal of the Korean Mathematical Society
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    • v.39 no.1
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    • pp.31-49
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    • 2002
  • An R$^{n}$ -geometry (P$^{n}$ , L) is a generalization of the Euclidean geometry on R$^{n}$ (see Def. 1.1). We can consider some topologies (see Def. 2.2) on the line set L such that the join operation V : P$^{n}$ $\times$ P$^{n}$ \ $\Delta$ longrightarrow L is continuous. It is a notable fact that in the case n = 2 the introduced topologies on L are same and the join operation V : P$^2$ $\times$ P$^2$ \ $\Delta$ longrightarrow L is continuous and open [10, 11]. It is a fundamental topological property of plane geometry, but in the cases n $\geq$ 3, it is no longer true. There are counter examples [2]. Hence, it is a fundamental problem to find suitable topologies on the line set L in an R$^{n}$ -geometry (P$^{n}$ , L) such that these topologies are compatible with the incidence structure of (P$^{n}$ , L). Therefore, we need to study the topologies of the line set L in an R$^{n}$ -geometry (P$^{n}$ , L). In this paper, the relations of such topologies on the line set L are studied.

Occurrence of Tn3 Sequence Upstream of aacC2 Gene in Gentamicin Resistance R Plasmids (Gentamicin 저항성 R 플라스미드에 존재하는 aacC2 유전자의 상류부위에서 Tn3의 출현)

  • 한효심;김남덕;이영종;이효연;정재성
    • Korean Journal of Microbiology
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    • v.33 no.3
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    • pp.165-169
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    • 1997
  • Two gentamicin resistance R plasmids, pGM5 and pGM6, containing aacC2 gene were selected from environmental isolates. The gentamicin resistance determinants of R plasmids were cloned into the BamHI site of pUC18. Restriction enzyme map of inserted region of recombinant plasmids, pSYS and pSY6, and PCR results indicated that Tn3 sequence was located upstream of gentamicin resistance gene. Based on the restriction maps and susceptibility tests, it was concluded that the sequence of bla and 3' inverted repeat of Tn3 play a important roles in the expression of gentamicin resistance gene.

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SR-ADDITIVE CODES

  • Mahmoudi, Saadoun;Samei, Karim
    • Bulletin of the Korean Mathematical Society
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    • v.56 no.5
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    • pp.1235-1255
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    • 2019
  • In this paper, we introduce SR-additive codes as a generalization of the classes of ${\mathbb{Z}}_{p^r}{\mathbb{Z}}_{p^s}$ and ${\mathbb{Z}}_2{\mathbb{Z}}_2[u]$-additive codes, where S is an R-algebra and an SR-additive code is an R-submodule of $S^{\alpha}{\times}R^{\beta}$. In particular, the definitions of bilinear forms, weight functions and Gray maps on the classes of ${\mathbb{Z}}_{p^r}{\mathbb{Z}}_{p^s}$ and ${\mathbb{Z}}_2{\mathbb{Z}}_2[u]$-additive codes are generalized to SR-additive codes. Also the singleton bound for SR-additive codes and some results on one weight SR-additive codes are given. Among other important results, we obtain the structure of SR-additive cyclic codes. As some results of the theory, the structure of cyclic ${\mathbb{Z}}_2{\mathbb{Z}}_4$, ${\mathbb{Z}}_{p^r}{\mathbb{Z}}_{p^s}$, ${\mathbb{Z}}_2{\mathbb{Z}}_2[u]$, $({\mathbb{Z}}_2)({\mathbb{Z}}_2+u{\mathbb{Z}}_2+u^2{\mathbb{Z}}_2)$, $({\mathbb{Z}}_2+u{\mathbb{Z}}_2)({\mathbb{Z}}_2+u{\mathbb{Z}}_2+u^2{\mathbb{Z}}_2)$, $({\mathbb{Z}}_2)({\mathbb{Z}}_2+u{\mathbb{Z}}_2+v{\mathbb{Z}}_2)$ and $({\mathbb{Z}}_2+u{\mathbb{Z}}_2)({\mathbb{Z}}_2+u{\mathbb{Z}}_2+v{\mathbb{Z}}_2)$-additive codes are presented.