• Archives of Pharmacal Research
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• v.27 no.8
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• pp.825-828
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• 2004

Two triterpenoids (1,4) and two triterpenoid glycosides (2,3) were isolated from the root of Acanthopanax koreanum (Araliaceae). Their structures were identified as impressic acid (1), acankoreoside A (2), 3-epi-betulinic acid 28-O-［(${\alpha}-L-rhamnopyranosyl(1{\rightarrow}4)-{\beta}-D-glucopyrano-syl(1{\rightarrow}6)]-{\beta}-D-glucopyranosyl]$ ester (3), and ursolic acid (4) by physicochemical and spectro-scopic methods. Of these compounds, impressic acid (1) exhibited a potent inhibitory activity against NFAT transcription factor ($IC_{50}:{\;}12.65{\;}{\mu\textrm{m}}$).

• Archives of Pharmacal Research
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• v.27 no.7
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• pp.738-741
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• 2004

Three lignans isolated from the roots of A. koreanum (Araliaceae), namely eleutheroside E(1), tortoside A(2), and hemiariensin(4), were evaluated for their ability to inhibit NFAT transcription factor. Of these compounds, compound 4, possessing a diarylbutane skeleton, exhibited potent inhibitory activity against NFAT transcription factor (($IC_{50}$ ： 36.3${\pm}2.5{\mu}\textrm{M}$). However, the activities of 1 (($IC_{50}$：＞500 11M) and 2 (($IC_{50}$： 136.1 ${\pm}9.4\mu\textrm{M}$), which possess bisaryldioxabicy-clooctane skeletons, were lower. As the lignan derivatives of the same skeletons, hinokinin (5) and (-)-yatein (6) with diarylbutane skeletons and(＋)-syringaresinol (3) with a bisaryldioxabicy-clooctane skeleton were also studied for their inhibitory effects on NFAT transcription factor.

• Journal of Applied Biological Chemistry
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• v.60 no.4
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• pp.301-306
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• 2017

This study was carried out to investigate the residual level of 5-methyl-1,2,4-triazolo[3,4-b][1.3] benzothiazole (tricyclazole) and the amount of transfer to Korean cabbage grown in treated soil with tricyclazole. The field trial on Korean cabbage was done at two different green houses located in Gwangju (Field 1) and Yongin (Field 2). Soil and cabbage samples were collected at different days after soil treatment of tricyclazole with two different concentration levels, respectively. Average recoveries of tricyclazole ranged from 83.5 to 92.1% in soil and cabbage and the variation coefficient was 1.3-6.8%. The initial concentrations of tricyclazole in field 1 soil were 4.25 and 8.97 mg/kg and decreased to 2.48 and 4.26 mg/kg at 43 DAT (day after treatment) and 0.88 and 2.02 mg/kg and decreased to 0.43 and 0.98 mg/kg at 36 DAT in field 2, respectively. The half-life of tricyclazole was about 39.6 and 28.1 days for the low and high concentration of tricyclazole treated soils in field 1 and 27.9 and 17.2 days for the low and high concentration of tricyclazole treated soils in field 2, respectively. Residual levels of tricyclazole in Korean cabbage were ranged from 4.03 to 18.26 and from 8.26 to 35.08% of initial concentration in filed 1 and field 2 soils, respectively.

• Journal of Bio-Environment Control
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• v.26 no.4
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• pp.235-241
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• 2017

This study was carried out to estimate growth characteristics of Kimchi cabbage cultivated in two different growing seasons and three transplanting dates in the greenhouses, and to create a predicting model for the production of Kimchi cabbage based on the growth parameters and climatic elements. Kimchi cabbages were transplanted three times at intervals of two weeks in spring and autumn growing seasons. Sigmoidal models for the estimation of fresh weight (Fw) was designed with days after transplanting, which were Fw=4451.5/[1+exp{-(DAT-34.1)/3.6}]($R^2=0.992$) and Fw=7182.0/[1+exp{-(DAT-53.8)/11.6}] ($R^2=0.979$), respectively. The relationship between fresh weight of Kimchi cabbage and growing degree days (GDD) was highly correlated, and the regression model represented by Fw=4451.5/[1+exp{-(GDD-34.1)/3.6}] ($R^2=0.992$) in spring growing season. The yield of Kimchi cabbage under spring and autumn growing season were estimated 11348.3kg/10a and 15128.2kg/10a, respectively, which were much different than outdoor culture each growing season, while greenhouse cultivation have shown similar results. To estimate the efficacy of prediction yield in Kimchi cabbage, we will need to supplement a predicting model, which was based on the parameters and climatic elements by the field cultivation.

• Archives of Pharmacal Research
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• v.28 no.6
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• pp.657-659
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• 2005

A new biflavonol glycoside named as solanoflavone (1) was isolated from aerial part of Solanum melongena. The chemical structure was elucidated as isorhamnetin-3-O-$\beta$-D-glucopyranoside-(4'$\to$O$\to$4"')-galangin-3"-O-$\to$-D-glucopyranoside on the basis of physicochemical and spectroscopic methods, including 2D NMR spectral techniques.

• Archives of Pharmacal Research
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• v.26 no.12
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• pp.1014-1017
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• 2003

Two new phenylpropanoid glycosides, 1-$\beta$-D-glucopyranosyl-2,6-dimethoxy-4-propenylphenol (1) and 1-[$\beta$-D-glucopyranosyl-(1$\rightarrow6)-\beta$-D-glucopyranosyl]-2,6-dimethoxy-4-propenylphenol (2) were isolated from the stem bark of Acanthopanax trifoliatus along with four known compounds (3∼6). Their structures were established on the basis of spectral and chemical evidences.

• Journal of the Korean Ceramic Society
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• v.44 no.7
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• pp.358-361
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• 2007

Well-ordered mesoporous SiCBN ceramics have been successfully synthesized by infiltrating a polymeric precursor, which was prepared from borazine and 2,4,6-trimethyl-2,4,6-trivinylcyclotrisilazane via a hydroboration reaction, into a mesoporous carbon (CMK-3) as a hard template. This was followed by pyrolysis at $1400^{\circ}C$ under nitrogen gas and subsequent oxidative removal of the carbon template without chemical etching. The prepared mesoporous SiCBN ceramic was characterized by a small-angle XRD, TEM, and BET surface area. The resulting mesoporous SiCBN ceramic revealed a BET surface area of $275 m^2g^{-1}$ and a pore volume of $0.8 cm^3 g$ with no crystallization.

• Journal of IKEEE
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• v.22 no.4
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• pp.948-952
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• 2018

Haze removal is an object of scientific desire due to its various practical applications. Existing algorithms are founded upon histogram equalization, contrast maximization, or the growing trend of applying machine learning in image processing. Since machine learning-based algorithms solve problems based on the data, they usually perform better than those based on traditional image processing/computer vision techniques. However, to achieve such a high performance, one of the requisites is a large and reliable training database, which seems to be unattainable owing to the complexity of real hazy and haze-free images acquisition. As a result, researchers are currently using the synthetic database, obtained by introducing the synthetic haze drawn from the standard uniform distribution into the clear images. In this paper, we propose the enhanced equidistribution, improving upon our previous study on equidistribution, and use it to make a new database for training machine learning-based haze removal algorithms. A large number of experiments verify the effectiveness of our proposed methodology.

• Journal of Applied Biological Chemistry
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• v.60 no.4
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• pp.343-349
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• 2017

This study was conducted to investigate the residual level and the amount of transfer to lettuce grown in field condition treated with the 5-methyl-1,2,4-triazolo[3,4-b][1,3]benzothiazole (Azoxystrobin). The field trials on lettuce were carried out at two different green houses located in Gwangju (Field 1) and Yongin (Field 2). Soil and lettuce samples were collected at different days after soil treatment of azoxystrobin with two different concentrations, respectively. Average recoveries for azoxystrobin ranged from 86.9 to 113.6% from soil and lettuce with the variation coefficient of 0.1-4.6%. The initial concentrations of azoxystrobin in Gwangju soil were 9.20, 11.00 mg/kg and decreased to 1.36, 2.70 mg/kg at 43 DAT (days after treatment) in field 1, while 1.06, 2.23 mg/kg decreased to 0.20 and 0.67 mg/kg at 36 DAT in field 2, respectively. The half-lives of azoxystrobin were about 19.4 and 23.3 days for the low and high concentration of azoxystrobin treated soils in field 1 and 11.5 and 17.8 days in field 2 soils, respectively. Residue levels of azoxystrobin in lettuce were not detected in filed 1 and field 2 soils, respectively.

• The Korean Journal of Pesticide Science
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• v.19 no.3
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• pp.174-184
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• 2015

In the present study, the metabolism of [$^{14}C$]butachlor was investigated in rice plant according to the OECD test guideline No. 501. [$^{14}C$]Butachlor was treated as granule to paddy water by application of 1.5 kg ingredient (a.i.)/ha at the 3~4 leave stage of rice plant. At 85 days after treatment (DAT), samples of panicle, foliage, and roots were taken for radioactivity analysis. Upon harvest at 126 DAT, rice plants were separated into brown rice, husk, straw, and root parts. Amounts of total radioactivity absorbed by rice plant ranged from 8.6 to 9.8% of applied radioactivity (AR). Total radioactive residues (TRRs) of rice plant at 126 DAT was the highest as 4.0421 mg/kg (7.3% AR) in the straw followed by 1.4595 mg/kg (2.4% AR) in the root, 0.7257 mg/kg (0.1% AR) in the husk. The lowest level recording 0.1020 mg/kg (0.1% AR) was found in brown rice. Each part was extracted with various solvents and solvent/water mixtures. Greater than 70% of TRRs was readily extractable from foliage, panicle, husk and straw. Only 34.0% of the brown rice and 43% of root based on TRRs were extractable showing that the residues were completely assimilated in the plant tissue. The level of non-extractable radioactivity was ranged from 26.2 to 66.0% of TRRs. From this study, five tentative major metabolites (M1, M2, M3, M4 and M5) were observed in rice extracts. Among the metabolites, 2,6-diethylaniline assigned as M4 was identified in rice plant by comparing to retention time of reference standard. Un-metabolized butachlor was not detected in any fractions. In soil extracts, N-(butoxymethyl)-N-(2,6-diethyl phenyl)acetamide, 2,6-diethylaniline, M2, M3 and M5 were observed. And the concentration of butachlor was low level (ca. 0.03 mg/kg).