1 |
Chien EY, Liu W, Zhao Q, Katritch V, Han GW, Hanson MA, et al. Structure of the human dopamine D3 receptor in complex with a D2/D3 selective antagonist. Science 2010;330:1091-1095.
DOI
|
2 |
Shimamura T, Shiroishi M, Weyand S, Tsujimoto H, Winter G, Katritch V, et al. Structure of the human histamine H1 receptor complex with doxepin. Nature 2011;475:65-70.
DOI
ScienceOn
|
3 |
Medina VA, Rivera ES. Histamine receptors and cancer pharmacology. Br J Pharmacol 2010;161:755-767.
DOI
ScienceOn
|
4 |
Schwartz JC, Arrang JM, Garbarg M, Pollard H, Ruat M. Histaminergic transmission in the mammalian brain. Physiol Rev 1991;71:1-51.
DOI
|
5 |
Hill SJ. Distribution, properties, and functional characteristics of three classes of histamine receptor. Pharmacol Rev 1990;42:45-83.
|
6 |
Hill SJ, Ganellin CR, Timmerman H, Schwartz JC, Shankley NP, Young JM, et al. International Union of Pharmacology. XIII. Classification of histamine receptors. Pharmacol Rev 1997;49:253-278.
|
7 |
Keller A, Vosshall LB. A psychophysical test of the vibration theory of olfaction. Nat Neurosci 2004;7:337-338.
DOI
ScienceOn
|
8 |
Takane SY, Mitchell JB. A structure-odour relationship study using EVA descriptors and hierarchical clustering. Org Biomol Chem 2004;2:3250-3255.
DOI
ScienceOn
|
9 |
Godden JW, Xue L, Bajorath J. Combinatorial preferences affect molecular similarity/diversity calculations using binary fingerprints and Tanimoto coefficients. J Chem Inf Comput Sci 2000;40:163-166.
DOI
ScienceOn
|
10 |
Schmidt MW, Baldridge KK, Boatz JA, Elbert ST, Gordon MS, Jensen JH, et al. General atomic and molecular electronic structure system. J Comput Chem 1993;14:1347-1363.
DOI
ScienceOn
|
11 |
Keseru GM, Makara GM. The influence of lead discovery strategies on the properties of drug candidates. Nat Rev Drug Discov 2009;8:203-212.
DOI
ScienceOn
|
12 |
Bleicher KH, Bohm HJ, Müller K, Alanine AI. Hit and lead generation: beyond high-throughput screening. Nat Rev Drug Discov 2003;2:369-378.
DOI
ScienceOn
|
13 |
Zheng CJ, Han LY, Yap CW, Ji ZL, Cao ZW, Chen YZ. Therapeutic targets: progress of their exploration and investigation of their characteristics. Pharmacol Rev 2006;58:259-279.
DOI
ScienceOn
|
14 |
Drews J. Drug discovery: a historical perspective. Science 2000;287:1960-1964.
DOI
|
15 |
Cherezov V, Rosenbaum DM, Hanson MA, Rasmussen SG, Thian FS, Kobilka TS, et al. High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor. Science 2007;318:1258-1265.
DOI
|