Effect of Additive of the Encapsulated Amounts and Solubility of Poorly Water-soluble Ibuprofen in Gelatin Microcapsules |
Li, Dong Xun
(College of Pharmacy, Yeungnam University)
Park, Jung-Gil (College of Pharmacy, Yeungnam University) Han, Hong-Hee (College of Pharmacy, Yeungnam University) Yang, Chan-Woo (College of Pharmacy, Yeungnam University) Choi, Jun-Young (College of Pharmacy, Yeungnam University) Oh, Dong-Hoon (College of Pharmacy, Yeungnam University) Yong, Chul-Soon (College of Pharmacy, Yeungnam University) Choi, Han-Gon (College of Pharmacy, Yeungnam University) |
1 | D.J. Germhalgh, A.C. Williams, P. Timmins and P. York, Solubility parameters as predictors of miscibility in solid dispersions, J. Pharm. Sci., 88, 1182-1190 (1999) DOI |
2 | L.C. Menting, B. Hoogstad and H.A.C. Thijssen, Diffusion coefficient of water and organic volatiles in carbohydratewater system, J. Food Technol., 5, 111-126 (1970) DOI |
3 | J. Sato and T. Kurusu, Process of manufacturing alcohol-containing solid matter, US Patent., 3786159 (1974) |
4 | J.S. Kaka and A. Tekle, Bioavailability of ibuprofen from oral and suppository preparations in rats, Res. Commun. Chem. Pathol. Pharmacol., 76, 171-182 (1992) |
5 | C.K. Kim, J.Y. Choi, Y.S. Yoon, J.P. Gong, H.G Choi, J.Y. Lee and B.J. Kong, Preparation and evaluation of dry elixir for the enhancement of dissolution rate of poorly water-soluble drugs, Int. J. Pharm., 106, 25-32 (1994) DOI ScienceOn |
6 | F.K. Glowka, Stereoselective pharmacokinetics of ibuprofen and its lysinate from suppositories in rabbits, Int. J. Pharm., 199, 159-166 (2000) DOI ScienceOn |
7 | J.L. Murtha and H.Y Ando, Synthesis of the cholesteryl ester prodrugs cholesteryl ibuprofen and cholesteryl flufenamate and their formulation into phospholipid microemulsions, J. Pharm. Sci., 83, 1222-1228 (1994) DOI ScienceOn |
8 | C.M. Adeyeye and J.C. Price, Development and evaluation of sustained-release ibuprofen-wax microspheres. 11. In vitro dissolution studies, Pharm. Res., 11, 575-579 (1994) DOI |
9 | A.K. Bansal, R.K. Khar, R. Dubey and A.K. Sharma, Effect of group substitution on the physicochemical properties of ibuprofen prodrugs, Pharmazie., 49, 422-424 (1994) |
10 | M. Charoenchaitrakool, F. Dehghani and N.R. Foster, Utilization of supercritical carbon dioxIGM for complex formation of ibuprofen and methyl-beta-cyclodextrin, Int. J. Pharm., 239, 103-112 (2002) DOI ScienceOn |
11 | L.C. Menting and B. Hoogstad, Volatile retention during the drying aqueous carbohydrate solutions, J. Food Sci., 32, 87-90 (1967) DOI |
12 | M.K. Ghorab and M.C. Adeyeye, Enhancement of ibuprofen dissolution via wet granulation with beta-cyclodextrin, Pharm. Dev. Technol., 6, 305-314 (2001) DOI ScienceOn |
13 | R. Bodmeier and J. Wang, Microencapsulation of drugs with aqueous colloidal polymer dispersions, J. Pharm. Sci., 82, 191-194 (1993) DOI |
14 | C.S. Yong, M.K. Lee, Y.J Park, K.H. Kong, J.J. Xuan, J.H. Kim, J.A. Kim, W.S. Lyoo, S.S. Han, J.O. Rhee, J.O. Kim, C.H. Yang, C.K. Kim and H.G Choi, Enhanced oral bioavailability of ibuprofen in rats by poloxamer gel using poloxamer 188 and menthol, Drug Dev. Ind. Pharm., 31, 615-622 (2005) DOI ScienceOn |
15 | S.W Lee, M.H. Kim and C.K. Kim, Encapsulation of ethanol by spray drying technique: effects of sodium lauryl sulfate, Int. J. Pharm., 187, 193-198 (1999) DOI ScienceOn |
16 | C.S. Yong, Y.K. Oh, S.H. Jung, J.D. Rhee, H.D. Kim, C.K. Kim, J.S. Choi and H.G Choi, Preparation of ibuprofen-loaded liquid suppository using eutectic mixture system with menthol, Eur. J. Pharm. Sci., 23, 347-353 (2004) DOI ScienceOn |
17 | H.J. Ahn, K.M. Kim and C.K. Kim, Enhancement of bioavailability of ketoprofen using drug elixir as a novel dosage form, Drug Dev. Ind Pharm., 24(7), 697-701 (1998) DOI |
18 | C.K. Kim and Y.S. Yoon, Developement of digoxin dry elixir as a novel dosage form using a spray-drying technique, J. Microencapsul., 12, 547-556 (1995) DOI |
19 | H.G Choi, B.J. Lee, C.S. Yong, J.D. Rhee, J.H. Han, M.K. Lee, K.M. Park and C.K. Kim, Terfenadine--cyclodextrin inclusion complex with the anti-histaminic activity enhancement, Drug Dev. Ind Pharm., 27, 857-862 (2001) DOI ScienceOn |
20 | G.M. Khan and Z. Jiabi, Ibuprofen release kinetics from controlled-release tablets granulated with aqueous polymeric dispersion of ethylcellulose II: Influence of several parameters and coexcipients, J. Controlled Rel., 56, 127-134 (1998) DOI ScienceOn |
21 | Z. Kokot and H. Zmidzinska, Solubility and dissolution rate of ibuprofen in ionic and non-ionic micellar systems, Acta Pol. Pharm., 58, 117-120 (2001) |
22 | C.S. Yong, C.H. Yang, J.D. Rhee, B.J. Lee, D.C. Kim, D.D. Kim, C.K. Kim, J.S. Choi and H.G. Choi, Enhanced rectal bioavailability of ibuprofen in rats by poloxamer 188 and menthol, Int. J. Pharm., 269, 169-176 (2004) DOI ScienceOn |
23 | C.K. Kim, Y.S. Yoon and lY Kong, Preparation and evaluation of flurbiprofen dry elixir as a novel dosage form using a spray-drying technique, Int. J. Pharm., 120,21-31 (1995) DOI ScienceOn |
24 | K. Kachrimanis, I. Nikolakakis and S. Malamataris, Spherical crystal agglomeration of ibuprofen by the solvent-change technique in presence ofmethacrylic polymers, J. Pharm. Sci., 89, 250-259 (2000) DOI ScienceOn |