Structure-Activity Relationship of 2-Substituted Hydroquinones as Tyrosinase Inhibitors for Topical Delivery |
Lee, Yeon-Jung
(College of Pharmacy, Pusan National University)
Yoon, Sung-Il (Dept. of Biotechnology, Dongseo University) Kim, Dae-Duk (College of Pharmacy and Research Institute of Pharmaceutical Sciences, Seoul National University) Kim, Jung-Sun (Dept. of Biotechnology, Dongseo University) |
1 | G. Negroiu, N. Branza-Nichita, A. J. Petrescu, T. A. Dwek and S. M. Petrescu, Protein specific N-glycosylation of tyrosinase and tyrosinase-related protein-1 in B16 mouse melanoma cells. Biochem. J., 344, 659-665 (1999) DOI ScienceOn |
2 | S. Bian, H-J. Doh, J. Zheng, J. S. Kim, C-H. Lee and D-D. Kim, In vitro evaluation of patch formulations for topical delivery of gentisic acid in rats, Eur. J. Pharm. Sci., 18, 141-147 (2003) DOI ScienceOn |
3 | S. Bian, J. Zheng, J. S. Kim, M. J. Choi, H-K. Chung, C-H. Lee and D-D. Kim, In vitro and in vivo studies of topical delivery system of gentisic acid in hairless mice, K. J. Pharm. Sci., 32, 161-164 (2002) |
4 | E. V. Curto, C. Kwong, H. Hermersdorfer, H. Glatt, C. Santis, V. Virador, V. J. Hearing and T. P. Dooley, Inhibitors of mammalian melanocyte tyrosinase: In Vitro comparisons of alkyl esters of gentisic acid with other putative inhibitors. Biochem. Pharmacol., 57, 663-672 (1999) DOI ScienceOn |
5 | J. J. Thiele, M. G Traber, T. G. Polefka, C. E. Cross and L. P. Packer, Ozone exposure depletes vitamin E and induces lipid peroxidation in murine stratum cormeum, J. Invest. Dermatol., 108, 753-757 (1997) DOI ScienceOn |
6 | M. Fontecave and J. L. Pierre, Oxidations by copper metallo-enzymes and some biomimetic approaches, Coordin. Chem. Rev., 170, 125-140 (1998) DOI ScienceOn |
7 | S. H. Pomerantz, Separation, purification, and properties of two tyrosinases from hamster melanoma, J. Biol. Chem., 238, 2351-2357 (1963) |
8 | T. Mosmann, Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays, J. Immunol. Methods., 65, 55-63 (1983) DOI ScienceOn |
9 | C. Hansch, A. Leo and D Hoekman, Exploring QSAR Hydrophobic, Electronic, and Steric Constents (1995) ACS Professional Reference Book |
10 | W. Siegrist and A. N. Eberle, In situ melanin assay for MSH using mouse B16 melanoma cells in culture, Anal. Biochem., 159, 191-197 (1986) DOI ScienceOn |
11 | D. H. Kim, J. S. Hwang, H. S. Baek, K. J. Kim and B. G Lee, Development of 5-[(3-Aminopropyl)phosphinooxyl]-2-(hydroxymethyl)-4H-pyran-4-one as a novel whitening agent, Chem. Pharm, Bull., 51(2), 113-116 (2003) DOI ScienceOn |
12 | J. Cabans, S. Chazarra and F. Gacia-Carmona, Kojic Acid, a cosmetic skin whitening agent, is a slow-binding inhibitor of catecholase activity of tyrosinase, J. Pharm. Pharmacol., 46, 982-985 (1994) DOI ScienceOn |