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http://dx.doi.org/10.5012/jkcs.2010.54.3.287

Novel Peracetylated N-Lactosyl-1,2,4-Thiadiazolidin-3-one Hydrochlorides: Synthesis and Antimicrobial Studies  

Dandale, Anvita S. (Dept. of Applied Chemistry, Faculty of Tech. & Engg., The M. S. University of Baroda)
Mangte, Dattatraya V. (P. G. Department of Chemistry, Shri Shivaji College)
Deshmukh, Shirish P. (P. G. Department of Chemistry, Shri Shivaji College)
Publication Information
Journal of the Korean Chemical Society / v.54, no.3, 2010 , pp. 287-290 More about this Journal
Abstract
In the present work we described oxidative cyclisation of peracetylated lactosyl carbamides with N-phenyl-S-chloro isothiocarbamoyl chloride and structural elucidation of novel peracetylated N-Lactosyl-1,2,4-Thiadiazolidin-3-one hydrochlorides. Antimicrobial activities of the title compounds were determined against bacteria S. aureus, E. coli, P. Vulgaris, P. Aeruginosa and fungi A. Niger, Penicillium.
Keywords
Peracetylated lactosyl carbamides; Isothiocarbamoyl chloride; Cyclisation; Peracetylated lactosyl thiadiazolidin-3-one; Synthesis; Antimicrobial activity;
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