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http://dx.doi.org/10.5012/jkcs.2010.54.01.059

Synthesis and Antimicrobial Screening of Some Fluorinated Azoles Containing (2-(6-Methyl-2-P-tolyl-lH-imidazo[1,2-a]pyridin-3-yl) Nucleus  

Shelke, Sharad (Department of Chemistry, S. S. G. M. College)
Salunkhe, Nilesh (Department of Chemistry, S. S. G. M. College)
Sangale, Sandeep (Department of Chemistry, S. S. G. M. College)
Bhalerao, Swapnil (Department of Chemistry, S. S. G. M. College)
Naik, Nilesh (Department of Chemistry, University of Pune)
Mhaske, Ganesh (Department of Chemistry, S. S. G. M. College)
Jadhav, Ranjana (Department of Chemistry, S. S. G. M. College)
Karale, Bhausaheb (Department of Chemistry, S. S. G. M. College)
Publication Information
Journal of the Korean Chemical Society / v.54, no.1, 2010 , pp. 59-64 More about this Journal
Abstract
The synthesis of a series of fluorinated thiadiazoles 3, triazoles 4 and oxadiazoles 5 are synthesized from thiosemicarbazides 2 containing (2-(6-methyl-2-p-tolyl-lH-imidazo[1,2-a]pyridin-3-yl nucleus. These reactions were carried out by conventional method as well as ultra sound irradiation method. All products have been characterized by IR, 1H NMR, MS study and screened for their antimicrobial activity.
Keywords
Fluorinated azoles; Triazoles; Thiadiazoles; Oxadiazoles; Ultrasound; Antibacterial activity;
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