Browse > Article
http://dx.doi.org/10.5012/bkcs.2012.33.2.721

Biological Evaluation and Molecular Docking Study of 3-(4-Sulfamoylphenyl)-4-phenyl-1H-pyrrole-2,5-dione as COX-2 Inhibitor  

Pham, Van Chung (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Shin, Ji-Sun (Department of Pharmaceutical Biochemistry and Department of Life and Nanopharmaceutical Science, College of Pharmacy, Kyung Hee University)
Choi, Min-Ji (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Kim, Tae-Woo (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Lee, Ki-Jae (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Kim, Kyung-Ju (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Huh, Geun (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Kim, Jung-Ahn (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Choo, Dong-Joon (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Lee, Kyung-Tae (Department of Pharmaceutical Biochemistry and Department of Life and Nanopharmaceutical Science, College of Pharmacy, Kyung Hee University)
Lee, Jae-Yeol (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
Publication Information
Bulletin of the Korean Chemical Society / v.33, no.2, 2012 , pp. 721-724 More about this Journal
Keywords
$PGE_2$ production; Anti-inflammatory; COX-2; Docking study; 1H-Pyrrole-2,5-dione;
Citations & Related Records
 (Related Records In Web of Science)
연도 인용수 순위
  • Reference
1 Gautam, R.; Jachak, S. M.; Kumar, V.; Mohan, C. G. Bioorg. Med. Chem. Lett. 2011, 21, 1612.   DOI   ScienceOn
2 Singh, P.; Bhardwaj, A.; Kaur, S.; Kumar, S. Eur. J. Med. Chem. 2009, 44, 1278.   DOI   ScienceOn
3 MVD 2010.4.2 for Windows in Molegro ApS.
4 Selinsky, B. S.; Gupta, K.; Sharkey, C. T.; Loll, P. J. Biochemistry 2001, 40, 5172.   DOI   ScienceOn
5 Wang, J. L; Limburg, D.; Graneto, M. J.; Springer, J.; Hamper, J. R.; Liao, S.; Pawlitz, J. L.; Kurumbail, R. G.; Maziasz. T.; Talley, J. J.; Kiefer, J. R.; Carter, J. Bioorg. Med. Chem. Lett. 2010, 20, 7159.   DOI   ScienceOn
6 Chandrasekharan, N. V.; Dai, H.; Roos, K. L.; Evanson, N. K.; Tomsik, J.; Elton, T. S.; Simmons, D. L. Proc. Natl. Acad. Sci. U.S.A. 2002, 99, 13926.   DOI   ScienceOn
7 Lee, S. H.; Kim, M. H.; Han, H. J. Am. J. Physiol. Cell Physiol. 2009, 297, C207.   DOI   ScienceOn
8 Watson, D. J.; Harper, S. E.; Zhao, P.-L.; Quan, H.; Bolognese, J. A.; Simon, T. J. Arch. Intern. Med. 2000, 160, 2998.   DOI   ScienceOn
9 Hawkey, C. J. Lancet 1999, 353, 307.   DOI   ScienceOn
10 Chan, F. K.; Hung, L. C.; Suen, B. Y.; Wu, J. C.; Lee, K. C.; Leung, V. K.; Hui, A. J.; To, K. F.; Leung, W. K.; Wong, V. W.; Chung, S. C.; Sung, J. J. N. Engl. J. Med. 2002, 347, 2104.   DOI   ScienceOn
11 McGettigan, P.; Henry, D. JAMA 2006, 296, 1633.   DOI   ScienceOn
12 Mason, R. P.; Walter, M. F.; McNulty, H. P.; Lockwood, S. F.; Byun, J.; Day, C. A.; Jacob, R. F. J. Cardiovasc. Pharmacol. 2006, 47, S7.   DOI   ScienceOn
13 Moon, J. T.; Jeon, J. Y.; Park, H. A.; Noh, Y. S.; Lee, K. T.; Kim, J.; Choo, D. J.; Lee, J. Y. Bioorg. Med. Chem. Lett. 2010, 20, 734.   DOI   ScienceOn
14 Yun, K. J.; Shin, J. S.; Choi, J. H.; Back, N. I.; Chung, H. G.; Lee, K. T. Int. Immunopharmacol. 2009, 9, 1323.   DOI   ScienceOn
15 Uddin, M. J.; Praveen Rao, P. N.; Knaus, E. E. Bioorg. Med. Chem. 2004, 12, 5929.   DOI   ScienceOn
16 Churchill, L.; Graham, A. G.; Shih, C.-K.; Pauletti, D.; Farina, P. R.; Grob, P. M. Inflammopharmacology 1996, 4, 125.   DOI   ScienceOn
17 Manivannan, E.; Chaturvedi, S. C. Bioorg. Med. Chem. 2011, 19,4520.   DOI   ScienceOn
18 Abdel-Aziz, A. A.; ElTahir, K. E.; Asiri, Y. A. Eur. J. Med. Chem. 2011, 46, 1648.   DOI   ScienceOn