Browse > Article
http://dx.doi.org/10.5012/bkcs.2003.24.11.1655

Chemoselective N-Benzenesulfonylation of Aliphatic Amines  

Kim, Ho-Kyun (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Park, Yong-Dae (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Kim, Jeum-Jong (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Lee, Me-Ho (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Chung, Hyun-A (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Kweon, Deok-Heon (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Cho, Su-Dong (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Yoon, Yong-Jin (Department of Chemistry and Research Institute of Life Sciences, Gyeongsang National University)
Publication Information
Bulletin of the Korean Chemical Society / v.24, no.11, 2003 , pp. 1655-1658 More about this Journal
Abstract
Chemoselective N-benzenesulfonylation of aliphatic amines using 2-(4-nitrobenzenesulfonyl)-4,5-dichloropyridazin-3(2H)-one (2) gave the corresponding 4-nitrobenzenesulfonamides in good or excellent yield. This method is a simple, mild and general procedure for the chemoselective N-benzenesulfonylation of aliphatic amines.
Keywords
Chemoselective N-benzenesulfonylation; 2-(4-Nitrobenzenesulfonyl)-4,5-dichloropyridazin-3-one; Pyridazinone;
Citations & Related Records

Times Cited By Web Of Science : 10  (Related Records In Web of Science)
Times Cited By SCOPUS : 8
연도 인용수 순위
1 Fukuyama, T.; Jow, C.-K.; Cheung, M. Tetrahedron Lett. 1995, 36, 6373.   DOI   ScienceOn
2 Bhatt, U.; Mohamed, N.; Just, G.; Roberts, E.Tetrahedron Lett. 1997, 38, 3679.   DOI   ScienceOn
3 Ibuka, T.; Mimura, N.;Aoyama, H.; Akaji, M.; Ohno, H.; Miwa, Y.; Taga, T.; Nakai, K.;Tamamura, H.; Fujii, N.; Yamamoto, Y. J. Org. Chem. 1997, 62,999.   DOI   ScienceOn
4 Wuts, P. G. M.; Northuis, J. M. Tetrahedron Lett. 1998,39, 3889.   DOI   ScienceOn
5 Weireb, S. M.; Demiko, D. M.; Lessen, T. A. Tetrahedron Lett.1986, 27, 2099.   DOI   ScienceOn
6 Malgres, P. E.; See, M. M.; Askin, D.; Reider,P. J. Tetrahedron Lett. 1997, 38, 5253.   DOI   ScienceOn
7 Sun, P.; Weinreb, S. M.;Shang, M. J. Org. Chem. 1997, 62, 8604.   DOI   ScienceOn
8 Nihei, K.−I.; Kato,M. J.; Yamane, T.; Palma, M. S.; Konno, K. Synlett 2001, 1167.
9 Fukuyama, T.; Cheung, M.; Jow, C. K.; Hidai, Y.; Kan, T.Tetrahedron Lett. 1997, 38, 5581.
10 Silveira, C. C.; Bernard, C.R.; Braga, A. L.; Kaufman, T. S. Synlett 2002, 907.
11 Kweon, D. H.; Kim, H. K.; Kim, J. J.; Chung, H.-A.; Lee, W. S.;Kim, S. K.; Yoon, Y. J. J. Heterocyclic Chem. 2002, 39,203.   DOI
12 Kang, Y. J.; Chung, H.-A.; Kim, J. J.; Yoon, Y. J. Synthesis 2002,733.
13 Green, T. W.; Wuts, P. G. M. Protective Groups in Organic Synthesis, 2nd ed.; Wiely: New York, 1991; pp 379-386.