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http://dx.doi.org/10.22643/JRMP.2018.4.2.99

211At and 211At-labeled radiopharmaceuticals for targeted alpha therapy  

Kang, Choong Mo (Division of Applied RI, Korea Institute of Radiological and Medical Sciences)
Lee, Kyo Chul (Division of Applied RI, Korea Institute of Radiological and Medical Sciences)
Lee, Yong Jin (Division of Applied RI, Korea Institute of Radiological and Medical Sciences)
Publication Information
Journal of Radiopharmaceuticals and Molecular Probes / v.4, no.2, 2018 , pp. 99-105 More about this Journal
Abstract
$^{211}At$ is an alpha emitting radionuclide, which can be produced using cyclotron with alpha beam. In addition, its strong linear energy transfer and iodine-like chemistry make that $^{211}At$ is one of the most attractive radionuclide in the field of targeted alpha therapy. In this review, production, labeling, and radiopharmaceuticals of $^{211}At$ will be discussed.
Keywords
$^{211}At$; Astatine; Targeted alpha therapy; Radiotherapy; Alpha particle;
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