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The NMR-data for the compound 6a:
$^{I}H$ NMR ($CDCl_{3}$ , 400MHz)$\delta$ =7.89 (s, 1H, NH), 4.79 (s, 1H, OH) 4.53 (ddd, J=5.96 hz,1H, CH-Lac), 4.46 (ddd, J=5.96 hz, 1H, CH-Lac), 3.88 (m, 2 H,$CH_2$ ), 3.47-3.44 (m, 1 H, CH-Lac), 2.90 (d, J=6.96 hz, 2H,$CH_2$ ), 2.70 (d, J=6.12hz, 2H,$CH_2$ ), 2.52-2.49 (m, 1H, CH-Lac), 2.10-2.08 (m, 1H, CH-Lac), 2.0 (s, 1H, NH), 1.65 (m, 2H,$CH_2$ ), 1.48-1.39 (m. 8H,$CH_2$ ); HRMS (CI) calcd for$C_{13}H_{24}N_2O_5S$ ($M^+$ + 1) 320.4100, found 320.4101 (Abbreviations: DIEA; diisopropyl ethylamine, HOBt, 1-hydroxybenzotriazole, BOP; benzotriazol-l-yl-oxy-tris(dimethylamino)phosphonium hexafluorophosphate, NMP; N-methyl-2-pyrrolidone, THF; tetrahydrofuran, and DMF; dimethylformamide)