• Bulletin of the Korean Chemical Society
• /
• 제24권8호
• /
• pp.1193-1196
• /
• 2003

Palladium-catalyzed heteroannulation of 2-amino-3-iodoquinoline derivatives and 1-trimethylsilyl internal alkynes provided highly regioselective pyrrolo[2,3-b]quinolines with trimethylsilyl group next to the nitrogen atom in the pyrrole ring.

• Bulletin of the Korean Chemical Society
• /
• 제19권6호
• /
• pp.667-671
• /
• 1998

A series of 1-aryl-lH-pyrazolo[4,3-c]quinolines and 2-aryl-2H-pyrazolo[4,3-c]quinolines are prepared by reacting 3-acyl-4-chloroquinolines in ethanol or 3-acyl-4(lH)-quinolone in acetic acid with appropriate hydrazines as possible anti-ulcer agents. A regiospecific synthesis of 1-aryl-lH-pyrazolo[4,3-c]quinolines is also achieved. The central pyridine ring could be easily reduced by catalytic hydrogenation.

• Bulletin of the Korean Chemical Society
• /
• 제23권4호
• /
• pp.541-542
• /
• 2002

• Bulletin of the Korean Chemical Society
• /
• 제31권3호
• /
• pp.704-707
• /
• 2010

• Bulletin of the Korean Chemical Society
• /
• 제26권12호
• /
• pp.2038-2040
• /
• 2005

• Bulletin of the Korean Chemical Society
• /
• 제26권6호
• /
• pp.1001-1004
• /
• 2005

• Bulletin of the Korean Chemical Society
• /
• 제26권8호
• /
• pp.1286-1288
• /
• 2005

• Bulletin of the Korean Chemical Society
• /
• 제31권12호
• /
• pp.3605-3610
• /
• 2010

In the present study, some quinoline derivatives have been synthesized like 8-methoxy-4-methyl-2-amino-(3'-chloro-2'-oxo-4'-substituted aryl-1'-azetidinyl)quinolines 8-12 and 8-methoxy-4-methyl-2-amino-(2'-substituted aryl-4'-oxo-1',3'-thiazolidin-3'-yl) quinolines 13-17 from 8-methoxy-4-methyl-2-(substituted arylidenyliminoamino)-quinolines 3-7. The structural assignments of these compounds were based on spectral (IR, $^1H$-NMR, Mass) and elemental (C, H, N) analysis. Further, these compounds were evaluated for antibacterial activity against various bacterial strains. Three compounds 10, 11 and 16 were found to exhibit potent antibacterial activity as compared to the standard drug amphicillin.

• Bulletin of the Korean Chemical Society
• /
• 제26권2호
• /
• pp.323-326
• /
• 2005

• Bulletin of the Korean Chemical Society
• /
• 제33권1호
• /
• pp.43-47
• /
• 2012

An efficient synthetic method for the preparation of quinolines through indium(III) chloride-catalyzed tandem addition-cyclization-oxidation reactions of imines with alkynes was developed. The processes can provide a diverse range of quinoline derivatives in good yields from simple imines and alkynes.