DOI QR코드

DOI QR Code

Non-Phosphopeptide Inhibitor for Lck SH2 Domain: Solid-Phase Synthesis and Structure Activity Relationship of Rosmarinic Acid Analogs

  • Published : 2003.05.20

Abstract

Keywords

References

  1. Cantley, L. C.; Auger, K. R.; Carpenter, C.; Duckworth, B.;Graziani, A.; Kappeller, R.; Soltoff, S. Cell 1991, 64, 241.
  2. Botfield, M. C.; Green, J. Ann. Rep. Med. Chem. 1995, 30, 227. https://doi.org/10.1016/S0065-7743(08)60937-9
  3. Garcia-Echeverria, C. Curr. Med. Chem. 2001, 13, 1589.
  4. Broadbridge, R. J.; Sharma, R. P. Current Drug Targets 2000, 1, 365. https://doi.org/10.2174/1389450003349074
  5. Beaulieu, P. L.; Cameron, D. R.; Ferland, J. M.;Gauthier, J.; Ghiro, E.; Gillard, J.; Gorys, V.; Poirier, M.;Rancourt, J.; Wernic, D.; Llinas-Brunet, M.; Betageri, R.;Cardozo, M.; Hickey, E. R.; Ingraham, R.; Jakes, S.; Kabcenell,A.; Kirrane, T.; Lukas, S.; Patel, U.; Proudfoot, J.; Sharma, R.;Tong, L.; Moss, N. J. Med. Chem. 1999, 42, 1757. https://doi.org/10.1021/jm980676t
  6. Morelock, M. M.; Ingraham, R. H.; Betageri, R.; Jakes, S. J. Med. Chem.1995, 38, 1309. https://doi.org/10.1021/jm00008a009
  7. Vu, C. B. Curr. Med. Chem. 2000, 10, 1081.
  8. Songyang, Z.; Shoelson, S. E.; Chaudhuri, M.; Gish, G.; Pawson, T.; Haser, W. G.; King, F.; Roberts, T.; Patnofsky, S.; Lechleider, R. J.; Neel, B. G.; Birge, B.; Cantley, L. C. Cell 1993, 72, 767. https://doi.org/10.1016/0092-8674(93)90404-E
  9. Hur, E. M.; Choi, B.; Park, C.; Lee, J.; Park, D.; Yun, Y.; Lee, K. H.; Oh, J. E.; Ahn, C. S.; Lee, H. S.; Ahn, J. S.; Jung, S. I. U.S. 6,140,363 October 31, 2000.
  10. Won, J.; Hur, E. M.; Hur, Y.; Park, S.; Kang, M.; Choi, Y.; Park,C.; Lee, K. H.; Yun, Y. Eur. J. Immunology 2003, 33, 870. https://doi.org/10.1002/eji.200323010
  11. Hu, B.; Messersmith, P. B. Tetrahedron Lett. 2000, 41, 5795. https://doi.org/10.1016/S0040-4039(00)00957-6
  12. Kaiser, E.; Colescott, R. L.; Bossinger, C. D.; Cook, P. I. Anal.Biochem. 1970, 34, 595. https://doi.org/10.1016/0003-2697(70)90146-6
  13. Gilmer, T.; Rodriguez, M.; Jordan, S.; Crosby, R.; Alligood, K.;Green, K.; Kimery, M.; Wagner, C.; Kinder, D.; Charifson, P.;Hassell, A. M.; Willard, D.; Luther, M.; Rusnak, D.; Sternbach, D.D.; Mehrotra, M.; Peel, M.; Shampine, L.; Davis, R.; Robbins, J.;Patel, I. R.; Kassel, D.; Burkhart, W.; Moyer, M.; Bradshaw, T.;Berman, J. J. Biol. Chem. 1994, 269, 31711.
  14. Eck, M. J.; Atwell, S. K.; Shoelson, S. E.; Harrison, S. C. Nature1994, 368, 764. https://doi.org/10.1038/368764a0

Cited by

  1. Design and synthesis of small chemical inhibitors containing different scaffolds for lck SH2 domain vol.13, pp.20, 2003, https://doi.org/10.1016/s0960-894x(03)00735-2
  2. Inhibitors of JAKs/STATs and the kinases: a possible new cluster of drugs vol.9, pp.6, 2003, https://doi.org/10.1016/s1359-6446(03)03014-9
  3. Is JAK3 a new drug target for immunomodulation-based therapies? vol.25, pp.11, 2003, https://doi.org/10.1016/j.tips.2004.09.008
  4. Development of Novel Small Chemical Inhibitors for Lck SH Domain with in vitro T-cell Inhibitory Activity vol.27, pp.9, 2003, https://doi.org/10.5012/bkcs.2006.27.9.1353