Archives of Pharmacal Research

  • 제25권3호
  • /
  • Pages.250-257
  • /
  • 2002
  • /
  • 0253-6269(pISSN)
  • /
  • 1976-3786(eISSN)
대한약학회 (The Pharmaceutical Society of Korea)
권호 표지

Synthesis and Antimicrobial Activity of New Substituted Anili-nobenzimidazoles

  • Nofal, Z.M. (Therapeutical Chemistry Dept., National Research Centre) ;
  • Fahmy, H.H. (Therapeutical Chemistry Dept., National Research Centre) ;
  • Mohamed, H.S. (Therapeutical Chemistry Dept., National Research Centre)
  • 발행 : 2002.06.01
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초록

A series of benzimidazole derivatives carrying different heterocycles such as 1,2,3-thiadiazole, 1,3,4-thiadiazole, thiazolidine, 2,3-dihydro-thiazole, 1,3,4-oxadiazole, semicarbazone and substituted thiosemi-carbazones were synthesized. Also a series of 1-methylbenzimidazole carrying hydroxy ethyl-amide, substituted sulfonyl hydrazide and benzoyl hydrazide from aminobenzoyl group at position 2 of 1-methylbenzimidazole were synthesized. The antimicrobial evaluation of some of the new compounds was carried out.

키워드

참고문헌

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