Archives of Pharmacal Research

The Pharmaceutical Society of Korea (대한약학회)
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Synthesis and In Vitro Cytotoxicity of 4-Alkyl- or 4-Arylaminosubstituted Cyclopenta[c]quinoline Derivatives

  • Published : 2001.10.01
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Abstract

Twelve 4-substituted cyclopenta[c]quinoline derivatives were synthesized and evaluated in vitro cytotoxicity against four human cancer cell lines (HOP62, SK-OV-3, MD-MB-468 and T-47D). The compounds 6c and 6e bearing p-anisidine and pyrrolidine side chain were more active than the others.

Keywords

References

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