INHIBITORY EFFECTS OF RAMULUS MORI EXTRACTS ON MELANOGENESIS

  • Kim, Jeong-Ha (R&D center, Coreana Cosmetics Co. Ltd., Cheonan) ;
  • Lee, Kang-Tae (R&D center, Coreana Cosmetics Co. Ltd., Cheonan)
  • Published : 1998.09.01

Abstract

13 develop an active agent for skin whitening, we examined the inhibitory effects of 285 plant extracts on tyrosinase activity and found some plant extracts have an ability to inhibit tyrosinase activity. Of these plant extracts, ramulus mori extracts showed the highest inhibiting activity on enzyme activity. From these results, we selected ramulus mori as a new active agent for skin whitening. $IC_{50}$/ of this extracts on tyrosinase activity is 12.48$\mu\textrm{g}$/m1. Also, ramulus mori extracts showed inhibitory activity on melanin synthesis in B-16 melanoma cells. We isolated active compound from ramulus mori extracts using various column chromatography and recrystalization and identified its chemical structure using Mass spectroscopy, IR and NMR analysis. So, it is identified as Mulberrin, a maior compound of ramutus mori and turned out that it has potent ability on tyrosinase inhibition. $IC_{50}$/ of this compound for tyrosinase activity is 0.5$\mu\textrm{g}$/ml. Also, this compound showed potent inhibitory activity on melanin synthesis in B-16 melanoma cells. This extracts was turned out to be safe in many safety tests.

Keywords

References

  1. Cosmetics & Toiletries v.111 Skin lighteners M. Masuda;T. Tejima;T. Suzuki;G. Imokawa
  2. Cosmetics & Toiletries v.107 Ultraviolet light and pigmentation of the skin J. M. Pawelek;A. K. Chakraborty;M. P. Osber;J. L. Bolognia
  3. Fragnance J. no.14 Melanocyte activation mechanism in UV pigmentation G. Imokawa
  4. Pigment Cell Research v.1 Induction of melanogenesis suppression : cellular pharmacology and mode of differential action Y. Mishima;S. Hatta;Y. Ohyama;M. Inazu
  5. J. Soc. Cosmet. Chem. v.42 In vitro effectiveness of several whitening cosmetic components in human melanocytes K. Maeda;M. Fukuda
  6. Fragnance J. no.14 Melanogenesis inhibitory effect of oil-soluble extract and its action mechanism T. Ikeda;T. Kambara
  7. International J. Cos. Sci v.19 no.4 Biological screening of 100 plant extracts for cosmetics use(Ⅰ) : inhibitory activities of tyrosinase and LOPA auto-oxidation K. T. Lee;B. J. Kim;J. H. Kim;M. Y. Heo;H. P. Kim
  8. Heterocycles v.12 no.10 On the structures of mulberrin, mulberrochromene, cyclomulberrin, and cyclomulberrochromene T. Nomura;T. Fukai
  9. CTFA Safety Testing Guideline The cosmetic, Toiletry, and Fragnance Association, Inc.
  10. Dermal toxicity, Assoc. Food and Drug Officials, US, Appraisal of the safety of chemicals in food, drugs, and cosmetics J. H. Draize
  11. J. Inv. Derm. v.52 The identification of contact allergens by animal assay the guinea-pig maximization tes B. Magnusson;A. M. Kligman
  12. Yale, J. Biol. Med. v.46 Quantitative measurement of melanin as tyrosinase equivalents and as weight of purified melanin A Oikawa;M. Nakayasu
  13. Annali Di Chimica v.80 Kinetic investigations on the double enzymic activity of the tyrosinase mush room A. Vanni;D. Gastaldi;G. Giunata