Journal of the Korean Chemical Society (대한화학회지)

Korean Chemical Society (대한화학회)
권호 표지

Synthesis of p-Acetamidobenzenesulfonamide Containing O, O'-Diethyl DL-1-Aminobenzylphosphonate and Their Derivatives

O, O'-Diethyl DL-1-Aminobenzylphosphonate와 그의 유도체들을 포함한 p-Acetamidobenzenesulfonamide의 합성

  • Young Suk Kim (Department of Chemical Engineering, College of Engineering) ;
  • Suk In Hong (Department of Chemical Engineering, College of Engineering) ;
  • Yong Joon Kim (Department of Chemical Engineering, College of Engineering)
  • 김영석 (高麗大學校 工科大學 化學工學科) ;
  • 홍석인 (高麗大學校 工科大學 化學工學科) ;
  • 김용준 (高麗大學校 工科大學 化學工學科)
  • Published : 1983.08.20

⟨ Previous Next ⟩

Abstract

Six new compounds of p-acetamidobenzenesulfonamides which contain O, O'-diethyl-1-aminobenzylphosphonate and their derivatives were prepared: O, O'-diethyl N-(p-acetamidobenzenesulfonyl) aminobenzylphosphonate, N-(p-acetamidobenzenesulfonyl) aminobenzylphosphonic acid, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl) glycyl] aminobenzylphosphonate, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-DL-alanyl] aminobenzylphosphonate, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-L-leucyl] aminobenzylphosphonate, and O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-L-phenylalanyl]aminobenzylphosphonate. All the compounds were obtained as white crystals and characterized by means of elemental analysis and infrared spectroscopy.

새로운 O, O'-diethyl-1-aminobenzylphosphonate와 그의 유도체들을 포함한 다음의 6가지의 p-acetamidobenzenesulfonamide를 합성하였다. O, O'-diethyl N-(p-acetamidobenzenesulfonyl) aminobenzylphosphonate, N-(p-acetamidobenzenesulfonyl) aminobenzylphosphonic acid, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl) glycyl] aminobenzylphosphonate, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-DL-alanyl] aminobenzylphosphonate, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-L-leucyl] aminobenzylphosphonate, O,O'-diethyl N-[N-(p-acetamidobenzenesulfonyl)-L-phenylalanyl]aminobenzylphosphonate. 모든 화합물은 흰색 결정으로 얻었으며 적외선 분광법과 원소분석으로 확인되었다.

Keywords

References

  1. Nature v.184 M. Horiguchi;Kantatsu
  2. Biochemistry v.1 J. S. Kettredge;E. Roberts;D. G. Simonsen
  3. Science v.144 L. D. Quin
  4. J. Biochem. (Tokyo) v.56 T. Hori;O. Itsaka;H. Inoue;K. Yamada
  5. Agr. Biol. Chem. v.29 M. Kantatsu;M. Horiguchi
  6. Nature v.262 S. G. Cull-Candy;J. F. Donnellan;R. W. James;G.G. Lunt
  7. Antibiotics and Chemotherapy v.3 J.D. Thayer;H.J. Magnuson;M.S. Gravatt
  8. Analytical Chemistry of Phosphorus Compounds M. Horiguchi;M. Hallman
  9. 한국영향학회지 v.2 김숙희;김용준;조정남
  10. Nature v.272 J. G. Allen;F. R. Atherson;M. J. Hall;C. H. Hassel;S. W. Holmes;R. W. Lambert;L. J. Nisbet;P. S. Ringrose
  11. J. Chem. Research v.41 A. Kotynsky;W. T. Stec
  12. Synthesis v.239 J. Lukszo;R. Tyka
  13. Tetrahedron Letter R. Tyka
  14. J. Org. Chem. v.39 G. H. Birum
  15. Synthesis P.G. Baralid;M. Guarner;F. Moroder;G. D. Pollini;D. Simoni
  16. J. Amer. Chem. Soc. v.60 H. G. Kollof
  17. Atti accad. Lincet, Classe sci. fis., mat. nat. v.28 F.P. Mazza;C. Migliadi
  18. C.A. v.33 F.P. Mazza;C. Migliadi
  19. U.S. Patent, 2,592,105 Sydney Archer
  20. Biol. Kutatointezat Munkui. v.15 Georgy Ivanovics, Mayer
  21. C.A. v.42 Georgy Ivanovics, Mayer
  22. Arch. Pharm. v.290 Hildegard Bangaz;Horst Bangaz
  23. Tetrahedron v.9 M. Frankel;P. Moses
  24. Sbornik statei obschchei Khim. v.2 A. V. Kirsanov;E.A. Abrazhanova
  25. Zhur. Obshchei khim. v.28 A. V. Kirsanov;N. L. Egorova
  26. C.A. v.52 A. V. Kirsanov;N. L. Egorova
  27. Kenkyusho Nempo v.12 Kozo Oyamada;Shoji Morimura;Takamine
  28. C.A. v.55 Kozo Oyamada;Shoji Morimura;Takamine
  29. U.S. Patent, 3,910,969 Franz, John E.
  30. U.S. Patent, 4,302,601 GailH. Birum
  31. The Examination of New Organic Compounds W. T. Smith;R.L. Shriner
  32. Ind. Eng. Chem. Anal. Ed. v.12 E. C. Wagner
  33. J. Amer. Chem. Soc. v.75 M. F. Chalmer;G. M. Kosolapoff
  34. Doklady. Akad. Nauk. USSR v.98 V. L. Ryzhkon;M. I. Kabachnik;L. M. Trasevich;T. Ya. Medved;H. A. Zeitlenok;N. K. Marchenk;V. A. Vagzhanova;E. F. Ulanova;Cheburkina
  35. Bull. of Korean Chem. Soc. v.1 S. I. Hong;Y. J. Kim
  36. J. Korean Chem. Soc. v.19 M. K. No;S. I. Hong;Y. J. Kim
  37. Synthesis v.1 Hans. R. Kricheldorf
  38. J. Org. Chem. v.26 Alexander W. Spears;Howard Tickelman